Nebivolol functions as a β-adrenergic receptor blocking agent. In individuals with extensive metabolism (representing most of the population) and at doses equal to or less than 10 mg, nebivolol exhibits preferential selectivity for β1 receptors. In poor metabolisers and higher doses, nebivolol inhibits both β1- and β2-adrenergic receptors. Nebivolol does not possess intrinsic sympathomimetic or membrane-stabilizing activity at concentrations relevant to therapeutic effects. At clinically significant doses, Nebivolol does not display α1-adrenergic receptor blockade activity. Various metabolites, including glucuronides, contribute to the β-blocking activity.
B. Pharm
B. Pharm, MSc.
Frequently asked questions
It starts showing its effects within a few hours after consumption.
Avoid usage if you experience an allergic reaction (hypersensitivity) to Nebivolol. It is advisable to seek advice from a doctor promptly.
Do not stop taking this medication without consulting your doctor, even if you feel healthy.
Consult your doctor before taking this medication if you have kidney or liver issues to ensure its safety and proper dosage.
This medication does not affect contraception.
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